Significance of Biotransformation of drug
Biotransformation of drugs encompasses several processes where drugs are converted into metabolites via biological systems like fungi, promoting eco-friendly drug development. Additionally, it involves chemical changes facilitated by metabolic processes, especially from gut microbiota. This process is crucial as it enables the metabolism of drugs, such as Adriamycin, into either active forms or safer alternatives within the body, highlighting its significance in pharmacology and drug safety.
Synonyms: Drug metabolism, Drug transformation, Xenobiotic metabolism, Metabolism of drug, Drug modification, Drug biotransformation
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The concept of Biotransformation of drug in scientific sources
Biotransformation of drug involves converting drugs into metabolites through biological systems, like fungi, and through metabolic processes by gut microbiota, promoting environmentally friendly drug development and altering substances chemically.
From: International Journal of Pharmacology
(1) Chloramphenicol can retard the biotransformation process of several drugs in different species.[1]